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Publications

Published in Top 10% journals in the field

MOUDRÝ, P., K. CHROMÁ, S. BURSAC, S. VOLAREVIC, J. BÁRTEK
RNA-interference screen for p53 regulators unveils a role of WDR75 in ribosome biogenesis. Cell Death and Differentiation. 2022, 29(3), 687-696, ISSN: 1350-9047, PMID: 34611297,
FANG, L., B. ZHU, Y. ZHAO, W. CHEN, Z. YANG, L. KERRIGAN, K. LANGEBACH, M. DE MARS, K. IDLER, H. JACOB, Y. ZHENG, Y. YU, E. JAEGER, G. SCHROTH, O. ABAAN, K. TALSANIA, J. LACK, T. SHEN, S. STANBOULY, B. TRAN, J. SHETTY, Y. KRIGA, D. MEERZAMAN, C. NGUYEN, V. PETITJEAN, M. SULTAN, M. CAM, M. MEHTA, T. HUNG, E. PETERS, R. KALAMEGHAM, S. SAHRAEIAN, M. MOHIYUDDI, T. GUO, L. YAO, L. SONG, H. LAM, J. DRÁBEK, P. VOJTA, R. MAESTRO, D. GASPAROTTO, S. KOKS, E. REIMANN, A. SCHERER, J. NORDLUND, U. LILJEDAHL, R. JENSEN, M. PIROOZNIA, Z. LI, C. XIAO, S. SHERRY, R. KUSKO, M. MOOS, E. DONALDSON, Z. TEZAK, B. NING, W. TONG, J. LI, P. DUERKEN-HUGHES, C. CATALANOTTI, S. MAHESHWARI, J. SHUGA, W. LIANG, J. KEATS, J. ADKINS, E. TASSONE, V. ZISMANN, T. MCDANIEL, J. TRENT, J. FOOX, D. BUTLER, C. MASON, H. HONG, C. WANG, W. XIAO, I. SOMATIC
Establishing community reference samples, data and call sets for benchmarking cancer mutation detection using whole-genome sequencing. Nature Biotechnology. 2021, 39(9), 1151-60, ISSN: 1087-0156, PMID: 34504347,
XIAO, W., L. FANG, Y. ZHAO, J. LACK, M. GUAN, B. ZHU, E. JAEGER, L. KERRIGAN, T. BLOMQUIST, T. HUNG, M. SULTAN, K. IDLER, A. SCHERER, R. KUSKO, M. MOOS, C. XIAO, S. SHERRY, O. ABAAN, W. CHEN, X. CHEN, J. NORDLUND, U. LILJEDAHL, R. MAESTRO, M. POLANO, J. DRÁBEK, P. VOJTA, S. KOKS, E. REIMANN, B. MADALA, T. MERCER, C. MILLER, H. JACOB, T. TRUONG, A. MOSHREFI, A. NATARAJAN, A. GRANAT, G. SCHROTH, R. KALAMEGHAM, E. PETERS, V. PETITJEAN, A. WALTON, T. SHEN, K. TALSANIA, C. VERA, K. LANGEBACH, M. DE MARS, J. HIPP, J. WILLEY, J. WANG, J. SHETTY, Y. KRIGA, A. RAZIUDDIN, B. TRAN, Y. ZHENG, Y. YU, M. CAM, P. JAILWALA, C. NGUYEN, D. MEERZAMAN, Q. CHEN, B. ERNEST, U. MEHRA, R. JENSEN, W. JONES, J. LI, B. PAPAS, M. PIROOZNIA, Y. CHEN, F. SEIFUDDIN, Z. LI, X. LIU, W. RESCH, J. WANG, L. WU, G. YAVAS, C. MILES, B. NING, W. TONG, C. MASON, E. DONALDSON, S. LABABIDI, L. STAUDT, Z. TEZAK, H. HONG, C. WANG
Toward best practice in cancer mutation detection with whole-genome and whole-exome sequencing. Nature Biotechnology. 2021, 39(9), 1141-50, ISSN: 1087-0156, PMID: 34504346,
POKORNÝ, J., D. OLEJNÍKOVÁ, I. FRYDRYCH, B. LIŠKOVÁ, S. GURSKÁ, S. BENICKÁ, J. ŠAREK, J. KOTULOVÁ, M. HAJDÚCH, P. DŽUBÁK, M. URBAN
Substituted dienes prepared from betulinic acid - Synthesis, cytotoxicity, mechanism of action, and pharmacological parameters. European Journal of Medicinal Chemistry. 2021, 224, 113706, ISSN: 0223-5234, PMID: 34311159,
MISTRÍK, M., Z. ŠKROTT, P. MULLER, A. PANACEK, L. HOCHVALDOVA, K. CHROMÁ, T. BUCHTOVÁ, V. VANDOVA, L. KVÍTEK, J. BÁRTEK
Microthermal-induced subcellular-targeted protein damage in cells on plasmonic nanosilver-modified surfaces evokes a two-phase HSP-p97/VCP response. Nature Communications. 2021, 12(1), 713, ISSN: 2041-1723, PMID: 33514738,
GONZALES, G., J. HODOŇ, A. KAZAKOVA, C. D´ACUNTO, P. KANOVSKY, M. URBAN, M. STRNAD
Novel pentacyclic triterpenes exhibiting strong neuroprotective activity in SH-SY5Y cells in salsolinol- and glutamate-induced neurodegeneration models. European Journal of Medicinal Chemistry. 2021, 213, 113168, ISSN: 0223-5234, PMID: 33508480,
VANDA, D., V. CANALE, S. CHAUMONT-DUBEL, R. KURCZAB, G. SATALA, K. P., M. KRAWCZYK, W. PIETRUS, K. BLICHARZ, E. PEKALA, A. BOJARSKI, P. POPIK, P. MARIN, M. SOURAL, P. ZAJDEL
Imidazopyridine-Based 5-HT 6 Receptor Neutral Antagonists: Impact of N1-Benzyl and N1-Phenylsulfonyl Fragments on Different Receptor Conformational States. Journal of Medicinal Chemistry. 2021, 64(2), 1180-1196, ISSN: 0022-2623, PMID: 33439019,
CReM: chemically reasonable mutations framework for structure generation. Journal of Cheminformatics. 2020, 12(1), 28, ISSN: 1758-2946, PMID: 33430959,
URBAN, M., V. ŠLACHTOVÁ, L. BRULÍKOVÁ
Small organic molecules targeting the energy metabolism of Mycobacterium tuberculosis. European Journal of Medicinal Chemistry. 2021, 212, 113139, ISSN: 0223-5234, PMID: 33422979,
KRAJČOVIČOVÁ, S., R. JORDA, D. VANDA, M. SOURAL, V. KRYŠTOF
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton's tyrosine kinase. European Journal of Medicinal Chemistry. 2020, 211, 113094, ISSN: 0223-5234, PMID: 33340912,